SOLUTION STRUCTURE OF MATRIX METALLOPROTEINASE 3 (MMP-3) IN THE PRESENCE OF 3-4'-CYANOBYPHENYL-4-YLOXY)-N-HDYDROXYPROPIONAMIDE (MMP-3 INHIBITOR VII)
GIPKWRKTHL TYRIVNYTPD LPKDAVDSAV EKALKVWEEV TPLTFSRLYE GEADIMISFA VREHGDDYPF DGPGNVLAHA YAPGPGINGD AHFDDDEQWT KDTTGTNLFL VAAHEIGHSL GLFHSANTEA LMYPLYHSLT DLTRFRLSQD DINGIQSLYG P
Polymer type: polypeptide(L)
Total | 1H | 15N | |
---|---|---|---|
All | 30.7 % (340 of 1106) | 20.0 % (189 of 943) | 92.6 % (151 of 163) |
Backbone | 65.1 % (310 of 476) | 49.2 % (160 of 325) | 99.3 % (150 of 151) |
Sidechain | 4.8 % (30 of 630) | 4.7 % (29 of 618) | 8.3 % (1 of 12) |
Aromatic | 1.9 % (2 of 104) | 2.0 % (2 of 101) | 0.0 % (0 of 3) |
Methyl | 6.7 % (6 of 89) | 6.7 % (6 of 89) |
1. MMP3
GIPKWRKTHL TYRIVNYTPD LPKDAVDSAV EKALKVWEEV TPLTFSRLYE GEADIMISFA VREHGDDYPF DGPGNVLAHA YAPGPGINGD AHFDDDEQWT KDTTGTNLFL VAAHEIGHSL GLFHSANTEA LMYPLYHSLT DLTRFRLSQD DINGIQSLYG PSolvent system 90% H2O/10% D2O, Pressure 1 atm, Temperature 298 K, pH 8
# | Name | Isotope labeling | Type | Concentration |
---|---|---|---|---|
1 | MMP3 | [U-98% 15N] | 1 mM | |
2 | H2O | 90 % | ||
3 | D2O | 10 % |